This five-day medicinal chemistry school will focus on most modern aspects associated with small molecule drug discovery, highlighting the methodologies and technologies supporting hit generation, lead finding and lead optimization campaigns.

The teaching content will be targeted at young scientists working in the area of medicinal chemistry, but also from flanking disciplines such as biochemistry, pharmacy, pharmacology, or biophysics from the pharmaceutical and biotech industry. Given the broad spectrum and the timeliness of scientific topics discussed, the course also provides a valuable opportunity for advanced medicinal chemists to get acquainted with most recent developments in, e.g., the medicinal chemistry of novel target families, novel compound classes, and most modern optimization paradigms. In addition, a number of Ph.D. students and postdocs will be able to attend to receive a broad overview on scientific disciplines involved in modern drug discovery.

The event will thematically be structured along key topics of strategic relevance for medicinal chemistry that will be presented by opinion leaders in the field. The teaching content will further be intensified by hands-on tutorials in which the theoretical learning’s can immediately be applied to real life problems of pre-clinical drug discovery.

Co-Chairmen

• Dr. Gerhard Müller, Gotham Therapeutics
• Prof. Dr. Beat Ernst, University of Basel

Organizers

• Dr. Gerhard Müller, Gotham Therapeutics
• Dr. Katarzyna Borsuk